BDBM360486 (1S,2S)-N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-pyridinyl)-4H-1,2,4-triazol-3-::US10221162, Example 824.0::US9845310, Example 824.0

SMILES COc1cccc(OC)c1-n1c(NS(=O)(=O)[C@H](C)[C@H](OC(C)C)c2cnc(C)cn2)nnc1-c1cccc(C)n1

InChI Key InChIKey=FMVCZUJFTVBQNZ-CLOONOSVSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 360486   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM360486((1S,2S)-N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-p...)
Affinity DataEC50:  0.470nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM360486((1S,2S)-N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-p...)
Affinity DataEC50:  0.470nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent