BDBM361394 3-(((3,3-difluoro- cyclobutyl) (methyl)amino)methyl)- N-(1H-pyrazolo[4,3-b] pyridin-3- yl)isothiazolo[4,5-b] pyridin-6-amine::US10221172, Example 52

SMILES CN(Cc1nsc2cc(Nc3n[nH]c4cccnc34)cnc12)C1CC(F)(F)C1

InChI Key InChIKey=PJRIZOJCPGAOHA-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 361394   

TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM361394(3-(((3,3-difluoro- cyclobutyl) (methyl)amino)methy...)
Affinity DataEC50:  334nMAssay Description:In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent