BDBM361403 3-((3,3-difluoropiperidin- 1-yl)methyl)-N-(1H- pyrazolo[4,3-b]pyridin-3- yl)isothiazolo[4,5-b] pyridin-6-amine::US10221172, Example 61

SMILES FC1(F)CCCN(Cc2nsc3cc(Nc4n[nH]c5cccnc45)cnc23)C1

InChI Key InChIKey=KVMSKMPPCZLMHB-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 361403   

TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM361403(3-((3,3-difluoropiperidin- 1-yl)methyl)-N-(1H- pyr...)
Affinity DataEC50:  55.9nMAssay Description:In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent