BDBM362927 2,5-Difluoro-4-{[(1R*,2R*)-2-phenylcyclohexyl]oxy}-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide::US9845313, Example 3

SMILES Fc1cc(c(F)cc1O[C@@H]1CCCC[C@@H]1c1ccccc1)S(=O)(=O)Nc1ncns1

InChI Key InChIKey=NKYGCXJKUCJEFU-RHSMWYFYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 362927   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM362927(2,5-Difluoro-4-{[(1R*,2R*)-2-phenylcyclohexyl]oxy}...)
Affinity DataIC50:  270nMAssay Description:Current record was obtained by an automated patch clamp system “IonWorks Quattro (Molecular Devices Corporation)” in Population Patch Clamp mode. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent