BDBM365170 6-methyl-4-(2-((1-methyl-1H- pyrazol-5-yl)amino)pyridin- 4-yl)-9-(2,2,2-trifluoroethyl)- 8,9-dihydro-1,2,2a1,6- tetraazabenzo[cd]azulen- 7(6H)-one::US10517878, Compound I-86::US10842799, I-86::US9867833, Compound I-86(S)
SMILES CN1c2cc(cc3nnc(C(CC(F)(F)F)CC1=O)n23)-c1ccnc(Nc2ccnn2C)c1
InChI Key InChIKey=FKAMZHMNVQECDN-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 365170
Affinity DataIC50: 212nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair