BDBM368817 (2R)-N-(4-dimethylaminophenyl)-2-methyl-4- [6-(4-pyridyl)-7H-pyrrolo[2,3-d]pyrimidin-4- yl]piperazine-1-carboxamide::US10227357, Compound P-0066
SMILES C[C@@H]1CN(CCN1C(=O)Nc1ccc(cc1)N(C)C)c1ncnc2[nH]c(cc12)-c1ccncc1
InChI Key
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 368817
Affinity DataKi: 500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair