BDBM369500 1-methyl-3-(2-(4-(((1R,2S)-2-phenylcyclopropyl)amino)piperidin-1-yl)ethyl)urea::US10233152, Example 38

SMILES O=C1N(CCN2CCC(CC2)N[C@@H]2C[C@H]2c2ccccc2)C(=O)c2ccccc12

InChI Key InChIKey=FJWIWTOAXUZITD-FCHUYYIVSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369500   

TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM369500(1-methyl-3-(2-(4-(((1R,2S)-2-phenylcyclopropyl)ami...)
Affinity DataIC50:  23nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent