BDBM369508 1-morpholino-3-phenyl-2-(4-(((1R,2S)-2-phenylcyclopropyl)amino)piperidin-1-yl)propan-1-one::US10233152, Example 46

SMILES O=C(C(Cc1ccccc1)N1CCC(CC1)N[C@@H]1C[C@H]1c1ccccc1)N1CCOCC1

InChI Key InChIKey=VCYHCWGZNIZFKP-LHJLODMPSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369508   

TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM369508(1-morpholino-3-phenyl-2-(4-(((1R,2S)-2-phenylcyclo...)
Affinity DataIC50:  58nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent