BDBM370591 US10238638, Example 20

SMILES COc1cc(OCc2csc(n2)-c2ccc(cc2)C(=O)N2CC[C@@H](CO)C2)c2sc(nc2c1)-c1cn2nc(sc2n1)C(C)(F)F

InChI Key InChIKey=WOWQTNNYHOIHLQ-MRXNPFEDSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 370591   

TargetPRKC apoptosis WT1 regulator protein(Homo sapiens (Human))
Universite De Montreal

US Patent
LigandPNGBDBM370591(US10238638, Example 20)
Affinity DataIC50:  1.20E+3nMAssay Description:The FLIPR assay is an exemplary in vitro assay for measuring the activity of the PAR4 antagonists of the present invention. In this assay, intracellu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent