BDBM371525 4-chloro-2-methyl-5-(((1R,3r,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl)amino)pyridazin-3(2H)-one::US10239861, Example 5
SMILES CN1[C@H]2CC[C@@H]1C[C@@H](C2)Nc1cnn(C)c(=O)c1Cl
InChI Key InChIKey=SQYCIYZYXUMJEO-ILWJIGKKSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 371525
Affinity DataIC50: 480nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair