BDBM371541 (racemic)-4-chloro-5-(((3RS,5SR)-1,5-dimethylpiperidin-3-yl)amino)-2-methylpyridazin-3(2H)-one::US10239861, Example 21
SMILES CC1CC(CN(C)C1)Nc1cnn(C)c(=O)c1Cl
InChI Key InChIKey=MRZBXPNVEWAIIA-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 371541
Affinity DataIC50: 36.5nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair