BDBM372513 N-[2-(4-Methyl-benzyl)-2H-[1,2,3]triazol-4-yl]-2-(1-methyl-1H-indazol-5-yl)-acetamide::US10246426, Example 69

SMILES Cc1ccc(Cn2ncc(NC(=O)Cc3ccc4n(C)ncc4c3)n2)cc1

InChI Key InChIKey=DZACNZJUPDJZBN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372513   

TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM372513(N-[2-(4-Methyl-benzyl)-2H-[1,2,3]triazol-4-yl]-2-(...)
Affinity DataIC50:  20nMAssay Description:Stock solutions of test compounds are prepared to a concentration of 10 mM in DMSO. For the Cav3.2 assay, serial dilutions of the compounds are prepa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent