BDBM375231 3-chloro-6-(5-fluoropyridin-3-yl)-5-(3-fluoropyridin-4-yl)pyridin-2-amine::US10253017, Example 27
SMILES Nc1cc(Cl)c(-c2ccnc(F)c2)c(n1)-c1cncc(F)c1
InChI Key InChIKey=YERBUXPLLAAXPI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 375231
Affinity DataKi: 150nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:The experiment of binding to MT3 sites was carried out on hamster brain membranes using [125I]2-iodomelatonin as radioligand in accordance with the p...More data for this Ligand-Target Pair