BDBM385539 3-(4-Chloro-2-hydroxy-3-methanesulfoximinophenylamino)-4-[(R)-1-(5-methylfuran-2-yl)propylamino]cyclobut-3-ene-1,2-dione::US10287278, Example 1

SMILES CC[C@@H](Nc1c(Nc2ccc(Cl)c(c2O)S(C)(=N)=O)c(=O)c1=O)c1ccc(C)o1

InChI Key InChIKey=OLLGDBDPMWUOJT-BKVLDKJMSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 385539   

TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM385539(3-(4-Chloro-2-hydroxy-3-methanesulfoximinophenylam...)
Affinity DataIC50: <200nMAssay Description:The in vitro affinity of the compounds of the present invention for the CXCR1 and CXCR2 receptors is determined on a functional test of β-arrest...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM385539(3-(4-Chloro-2-hydroxy-3-methanesulfoximinophenylam...)
Affinity DataIC50: <20nMAssay Description:The in vitro affinity of the compounds of the present invention for the CXCR1 and CXCR2 receptors is determined on a functional test of β-arrest...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent