BDBM389841 4-{5-[3-(4-Chlorophenyl)-3H- imidazo[4,5-c]pyridin-2- yl]pyrimidin-2-yl}piperazin-2- one::US10766897, Compound 13::US10968223, Compound 13::US9951068, Compound 13
SMILES Clc1ccc(cc1)-n1c(nc2ccncc12)-c1cnc(nc1)N1CCNC(=O)C1
InChI Key InChIKey=QBJRIEOQHPSKCT-UHFFFAOYSA-N
Data 7 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 389841
Affinity DataIC50: <50nMAssay Description:SSAO: All primary assays were performed at RT. with purified recombinantly expressed human SSAO. Enzyme was prepared essentially as described in Öhma...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Compounds of the invention were tested for inhibition of the human ether a go-go related gene (hERG) K+ channel using IonWorks patch clamp electrophy...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:All primary assays were performed at RT. with purified recombinantly expressed human SSAO. Enzyme was prepared essentially as described in Öhman et a...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:All primary assays were performed at RT. with purified recombinantly expressed human SSAO. Enzyme was prepared essentially as described in Öhman et a...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:SSAO: All primary assays were performed at RT. with purified recombinantly expressed human SSAO. Enzyme was prepared essentially as described in Öhma...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:hERG: Compounds of the invention were tested for inhibition of the human ether a go-go related gene (hERG) K+ channel using IonWorks patch clamp elec...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Electrophysiological recordings were made from a Chinese Hamster Lung cell line stably expressing the full length hERG channel. Single cell ion curre...More data for this Ligand-Target Pair