BDBM391796 5-((7-(4-Cyano-3-(trifluoromethyl)phenyl)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)amino)-N-(2,2-difluoroethyl)picolinamide::US10300067, Example 48

SMILES FC(F)CNC(=O)c1ccc(Nc2ncnc3CN(CCc23)c2ccc(C#N)c(c2)C(F)(F)F)cn1

InChI Key InChIKey=YKLABHRBKMZJRH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 391796   

TargetAndrogen receptor(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM391796(5-((7-(4-Cyano-3-(trifluoromethyl)phenyl)-5,6,7,8-...)
Affinity DataIC50:  490nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent