BDBM395249 US10308629, Example 11::rel-(4aR,7aS)-6-Methyl-3-(phenylamino)-2-(pyridin-4-yl)-1,4a,5,6,7a,8-hexahydropyrrolo[3,4-f]indole-4,7-dione
SMILES COC(=O)C1CC(O)=C(C(=S)Nc2ccccc2)C(=O)C1
InChI Key InChIKey=YJLNQXRRJGTRBC-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 395249
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft
US Patent
Bayer Pharma Aktiengesellschaft
US Patent
Affinity DataIC50: 19nMAssay Description:Bub1-inhibitory activities of compounds described in the present invention were quantified using a time-resolved fluorescence energy transfer (TR-FRE...More data for this Ligand-Target Pair