BDBM401240 US10005756, Compound A1

SMILES O[C@@]1(CCN(C1=O)c1cccc(c1)S(=O)(=O)N1CCNCC1)C(=O)NCc1cc(F)cc(Cl)c1

InChI Key InChIKey=MNYBMTDDNABXQH-QFIPXVFZSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 401240   

TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM401240(US10005756, Compound A1)
Affinity DataIC50:  130nMAssay Description:The MetAP-2 activity is determined by coupling enzymatic reactions. The tripeptide Met-Arg-Ser (MAS) is employed as substrate. The methionine liberat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent