BDBM402575 N-(4-cyanothiophen-3-yl)- 2-(1,4-diazepan-1- yl)pyrrolo[2,1- f][1,2,4]triazine-7- carboxamide trifluoroacetate::US10329295, Example 12
SMILES O=C(Nc1cscc1C#N)c1ccc2cnc(nn12)N1CCCNCC1
InChI Key InChIKey=MOSCEAKEAHUAKV-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 402575
Affinity DataIC50: 365nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair