BDBM402782 2-{[(1R,2R)-2-amino-3,3- difluorocyclohexyl]amino}- N-(3-bromo-1-methyl- 1H-pyrazol-4- yl)pyrrolo[2,1- f][1,2,4]triazine-7- carboxamide trifluoroacetate::US10329295, Example 89
SMILES Cn1cc(NC(=O)c2ccc3cnc(N[C@@H]4CCCC(F)(F)[C@@H]4N)nn23)c(Br)n1
InChI Key InChIKey=AWPFBQFOVUDWNE-ZWNOBZJWSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 402782
Affinity DataIC50: 373nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair