BDBM402792 2-[(1S,5S)- or (1R,5R)-3,6- diazabicyclo[3.2.1]oct-3- yl]-N-[1-methyl-3- (trifluoromethyl)-1H- pyrazol-4-yl]pyrrolo[2,1- f][1,2,4]triazine-7- carboxamide::US10329295, Example 100
SMILES Cn1cc(NC(=O)c2ccc3cnc(nn23)N2C[C@@H]3CN[C@@H](C3)C2)c(n1)C(F)(F)F
InChI Key InChIKey=OGXDDAVKGVTLEM-QWRGUYRKSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 402792
Affinity DataIC50: 64nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair