BDBM402810 N-(3-cyano-1-methyl-1H- pyrazol-4-yl)-2-{[(1R,2S)- 2- hydroxycyclohexyl]amino}- pyrrolo[2,1- f][1,2,4]triazine-7- carboxamide trifluoroacetate::US10329295, Example 122
SMILES Cn1cc(NC(=O)c2ccc3cnc(N[C@@H]4CCCC[C@@H]4O)nn23)c(n1)C#N
InChI Key InChIKey=FSRRITQUZUGHBF-WBMJQRKESA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 402810
Affinity DataIC50: 20nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair