BDBM404765 1-{4-[4-({1-[3- (trifluoromethoxy)phenyl]ethyl} carbamoyl)-1H-1,2,3-triazol-1-yl] butyl}-N-{[4-(trifluoromethyl) pyridin-2-yl]methyl}-1H-1,2,3- triazole-4-carboxamide::US10344025, Example 109::US11370786, Example 109
SMILES CC(NC(=O)c1cn(CCCCn2cc(nn2)C(=O)NCc2cc(ccn2)C(F)(F)F)nn1)c1cccc(OC(F)(F)F)c1
InChI Key InChIKey=ZEHJUNWJGNDYNH-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 404765
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board Of Regents, The University Of Texas System
US Patent
Board Of Regents, The University Of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board Of Regents, The University Of Texas System
US Patent
Board Of Regents, The University Of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair