BDBM405643 US10351547, Compound 2-61::US10597377, Compound 2-61

SMILES CO[C@H]1CN(CC[C@H]1N)c1c(cnc2ccc(cc12)-c1cccc(C#N)c1O)-c1cc(F)cc(F)c1

InChI Key InChIKey=IBYBYCAQCXHPOP-RSXGOPAZSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 405643   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM405643(US10351547, Compound 2-61 | US10597377, Compound 2...)
Affinity DataEC50:  55nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC # CCL-61) stably expressing the human SSTR2 are plated in each well of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM405643(US10351547, Compound 2-61 | US10597377, Compound 2...)
Affinity DataEC50:  55nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent