BDBM406619 5-(2,6- dimethoxyphenyl)- 6-(ethoxymethyl)- 3-(5- {[1,2]oxazolo[4,5- b]pyridin-3- ylmethyl}-1,3,4- oxadiazol-2- yl)pyridine-2,4-diol::US10336739, Example 228

SMILES CCOCc1nc(O)c(-c2nnc(Cc3noc4cccnc34)o2)c(O)c1-c1c(OC)cccc1OC

InChI Key InChIKey=UQQXSRJGLQXUQN-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 406619   

TargetApelin receptor(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM406619(5-(2,6- dimethoxyphenyl)- 6-(ethoxymethyl)- 3-(5- ...)
Affinity DataEC50:  5.5nMAssay Description:HEK293 cells stably expressing human APJ receptor were used to assess the activity of compounds. Cultured cells were detached and resuspended in the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent