BDBM412258 (5R,6S)-5-(4-((2-(3- (fluoromethyl)azetidin- 1- yl)ethyl)amino)phenyl)- 6-phenyl-5,6,7,8- tetrahydronaphthalen- 2-ol::US10399939, Example 137

SMILES Oc1ccc2[C@H]([C@H](CCc2c1)c1ccccc1)c1ccc(NCCN2CC(CF)C2)cc1

InChI Key InChIKey=NSYIAMPCRNXEOC-IAPPQJPRSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412258   

TargetEstrogen receptor(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM412258((5R,6S)-5-(4-((2-(3- (fluoromethyl)azetidin- 1- yl...)
Affinity DataEC50:  186nMAssay Description:The relative efficacies of Formula I compounds as inhibitors of an enzyme activity (or other biological activity) can be established by determining t...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent