BDBM412508 (E)-5-fluoro-4-methyl-N-(5-(1-(6- (pyrrolidin-1-yl)pyridin-3-yl)prop-1- en-1-yl)pyridin-2-yl)nicotinamide::US10399967, Compound 141

SMILES C\C=C(/c1ccc(NC(=O)c2cncc(F)c2C)nc1)c1ccc(nc1)N1CCCC1

InChI Key InChIKey=PUIWXZWHXRVFJB-QBROUFQSSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412508   

TargetInterleukin-2(Homo sapiens (Human))
Prcl Research

US Patent
LigandPNGBDBM412508((E)-5-fluoro-4-methyl-N-(5-(1-(6- (pyrrolidin-1-yl...)
Affinity DataIC50:  135nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent