BDBM420056 (S)-N-((1-isopropylpyrrolidin-2-yl)methyl)-10- methyl-1-oxo-2-(pyridin-3-yl)-1,2- dihydropyrazino[1,2-a]indole-4-carboxamide::US10487087, Compound 20

SMILES CC(C)N1CCC[C@H]1CNC(=O)c1cn(-c2cccnc2)c(=O)c2c(C)c3ccccc3n12

InChI Key InChIKey=GZXVAACFIKKZFS-FQEVSTJZSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 420056   

TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Vanderbilt University

US Patent

LigandBDBM420056((S)-N-((1-isopropylpyrrolidin-2-yl)methyl)-10- met...)Copy SMILESCopy InChI

Affinity DataEC50:  5.20E+3nMAssay Description:To assess the effects of test compounds on GLP-1 or glucagon potency and efficacy, a high-throughput calcium mobilization assay was used essentially ...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand Info

In DepthDetails US Patent
Copy BDB DOI