BDBM432157 N-(1-Benzylpiperidin-4-yl)-5-chloro-N-(1-phenyl-1H-pyrazol-3-yl)thiophene-2-::US10577360, Example 23
SMILES Clc1ccc(s1)C(=O)N(C1CCN(Cc2ccccc2)CC1)c1ccn(n1)-c1ccccc1
InChI Key InChIKey=KCFATVFDJGUCIV-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 432157
Affinity DataKi: 300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Esteve Pharmaceuticals
US Patent
Esteve Pharmaceuticals
US Patent
Affinity DataKi: >5.00E+3nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair