BDBM434777 US10562910, Example 4
SMILES OC(=O)c1cc(F)c2CCc3nc(OCc4c(onc4-c4c(Cl)cccc4Cl)C4CC4)ccc3Oc2c1
InChI Key InChIKey=ACQLAZWSLWBDRC-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 434777
TargetBile acid receptor(Homo sapiens (Human))
Southern Medical University Biomedical Research Center
Curated by ChEMBL
Southern Medical University Biomedical Research Center
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Agonist activity at human FXR expressed in HEK293T cells by luciferase reporter assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Southern Medical University Biomedical Research Center
Curated by ChEMBL
Southern Medical University Biomedical Research Center
Curated by ChEMBL
Affinity DataEC50: 60.4nMAssay Description:Purchasing invitrogen PV4833 kits. The procedure refers to LanthaScreen TR-FRET Farnesoid X Receptor Coactivator AssayFirst, the required amount of t...More data for this Ligand-Target Pair