BDBM434882 N-(2-Ethylbutyl)-N-(2-(pyridin-4-yl)ethyl)-4-(4-(trifluoromethoxy)phenyl)-1H-1,2,3-triazole-1-carboxamide::US10583137, Compound 53

SMILES CCC(CC)CN(CCc1ccncc1)C(=O)n1cc(nn1)-c1ccc(OC(F)(F)F)cc1

InChI Key InChIKey=PTACIMLVHPESHV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434882   

TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434882(N-(2-Ethylbutyl)-N-(2-(pyridin-4-yl)ethyl)-4-(4-(t...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434882(N-(2-Ethylbutyl)-N-(2-(pyridin-4-yl)ethyl)-4-(4-(t...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent