BDBM434893 (2-(pyridin-4- ylmethyl)piperidin-1-yl)(4- (2',4',6'-trimethoxy-[1,1'- biphenyl]-4-yl)-1H-1,2,3-triazol- 1-yl)methanone::US10583137, Compound 67

SMILES COc1cc(OC)c(c(OC)c1)-c1ccc(cc1)-c1cn(nn1)C(=O)N1CCCCC1Cc1ccncc1

InChI Key InChIKey=JJKGHTDXLZCXAH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434893   

TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434893((2-(pyridin-4- ylmethyl)piperidin-1-yl)(4- (2',4',...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434893((2-(pyridin-4- ylmethyl)piperidin-1-yl)(4- (2',4',...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent