BDBM434911 (2-benzylpiperidin-1-yl)(4- (2,4,6-trimethoxyphenyl)-1H- 1,2,3-triazol-2-yl)methanone::US10583137, Compound 85

SMILES COc1cc(OC)c(-c2cnn(n2)C(=O)N2CCCCC2Cc2ccccc2)c(OC)c1

InChI Key InChIKey=QRSBFGGXIOVBBR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434911   

TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434911((2-benzylpiperidin-1-yl)(4- (2,4,6-trimethoxypheny...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434911((2-benzylpiperidin-1-yl)(4- (2,4,6-trimethoxypheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent