BDBM435359 (trans)-N-((2-(2-hydroxy-2- methylpropanoyl)-5-(3- (trifluoromethyl)phenyl)-1,2,3,4- tetrahydroisoquinolin-8-yl)methyl)-2-(3- methyl-1,2,4-oxadiazol-5- yl)cyclopropanecarboxamide (mixture of 2 isomers)::US10568876, Example 120
SMILES Cc1noc(n1)[C@@H]1C[C@H]1C(=O)NCc1ccc(-c2cccc(c2)C(F)(F)F)c2CCN(Cc12)C(=O)C(C)(C)O
InChI Key InChIKey=JSPBEIZSGUUVPW-FGZHOGPDSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 435359
Affinity DataIC50: 1.58E+3nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product triolein (1,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membrane prep m...More data for this Ligand-Target Pair