BDBM437503 2-[4-(1'-Methyl-6'-oxo-1',6'-dihydro-[3,4']bipyridinyl-3'- yl)-pyrazol-1-yl]-benzonitrile::US10617680, Example 237::US11020380, Example 237

SMILES Cn1cc(-c2cnn(c2)-c2ccccc2C#N)c(cc1=O)-c1cccnc1

InChI Key InChIKey=UMSUTJZINTUCEA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437503   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437503(2-[4-(1'-Methyl-6'-oxo-1',6'-dihydro-[3,4']bipyrid...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437503(2-[4-(1'-Methyl-6'-oxo-1',6'-dihydro-[3,4']bipyrid...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent