BDBM439157 US10604514, Compound 33
SMILES Cc1nnc(s1)-c1ccc2cnc(NC(=O)N3CC[C@H](N)[C@@H](F)C3)cc2c1
InChI Key InChIKey=BFNNBSKNGPXKKS-GJZGRUSLSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 439157
Affinity DataEC50: 23nMAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed
US Patent
Samumed
US Patent
Affinity DataEC50: 9nMAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 _...More data for this Ligand-Target Pair