BDBM447765 US10689367, Example 136.0::US10689367, Example 86.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc(-c2ccccn2)n1C(C)C)c1ncc(Cl)cn1

InChI Key InChIKey=OTASHMRLTCCRMR-WFASDCNBSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 447765   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM447765(US10689367, Example 136.0 | US10689367, Example 86...)
Affinity DataEC50:  57nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM447765(US10689367, Example 136.0 | US10689367, Example 86...)
Affinity DataEC50:  57nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent