BDBM449028 US10702498, Compound 2::US11484525, Compound 2
SMILES C[NH+](C)[C@H](CNC(=O)Cc1cn2ccccc2n1)Cc1ccccc1
InChI Key InChIKey=PXBWXTKSXXKPTL-SFHVURJKSA-O
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 449028
TargetMu-type opioid receptor(Homo sapiens (Human))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 5.80E+3nMAssay Description:Each compound was initially tested at 20 μM and was incubated with 3H-DPN at a concentration equal to the Kd (0.4 nM) of the radioligand in _...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 5.80E+3nMAssay Description:For a primary screen of selected molecules, binding to μOR was assessed by measuring competition against the radioligand 3H-diprenorphine (3H-DPN). ...More data for this Ligand-Target Pair