BDBM458286 US10752616, Code No. BHBA-044

SMILES Cc1ccc(C)c2oc(cc12)-c1nsc(n1)-c1ccc(C(O)=O)c(F)c1

InChI Key InChIKey=BBSGLOXGWJXZPN-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 458286   

TargetRetinoic acid receptor beta(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458286(US10752616, Code No. BHBA-044)
Affinity DataEC50:  2nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458286(US10752616, Code No. BHBA-044)
Affinity DataEC50:  3.40nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458286(US10752616, Code No. BHBA-044)
Affinity DataEC50:  26nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent