BDBM4855 1-(4-Chloroanilino)-4-(3-pyridylmethyl)phthalazine Hydrochloride::CGP79787 Analog 40::N-(4-chlorophenyl)-4-(pyridin-3-ylmethyl)phthalazin-1-amine

SMILES Clc1ccc(Nc2nnc(Cc3cccnc3)c3ccccc23)cc1

InChI Key InChIKey=GNNTUYLPJHMKJZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4855   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM4855(1-(4-Chloroanilino)-4-(3-pyridylmethyl)phthalazine...)
Affinity DataIC50: >1.00E+4nMAssay Description:The in vitro kinase assays were performed in 96-well plates using the recombinant GST-fused kinase domains expressed in baculovirus and purified over...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM4855(1-(4-Chloroanilino)-4-(3-pyridylmethyl)phthalazine...)
Affinity DataIC50:  9.80E+3nMpH: 7.5 T: 2°CAssay Description:The in vitro kinase assays were performed in 96-well plates using the recombinant GST-fused kinase domains expressed in baculovirus and purified over...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed