BDBM50000570 3-(2-Methyl-2-aza-bicyclo[3.3.1]non-5-yl)-phenol::CHEMBL285250
SMILES CN1CCC2(CCCC1C2)c1cccc(O)c1
InChI Key InChIKey=ZQJGRSYDDMBMPJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 17 hits for monomerid = 50000570
Affinity DataKi: 3.40nMAssay Description:Binding affinity towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity of the compound towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Binding affinity of the compound towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity of the compound towards opioid receptor kappa 2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity of the compound towards opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: >500nMAssay Description:Binding affinity of the compound towards opioid receptor mu 2More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of [3H]DAMGO radioligand binding to rat brain opioid receptor mu 1.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of [3H]DAMGO radioligand binding to rat brain opioid receptor mu 1.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 911nMAssay Description:Inhibition of [3H]U-69593 radioligand binding to Guinea pig opioid receptor kappa 1.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 557nMAssay Description:Opioid activity against delta-receptor of isolated mouse vas deferens(MVD) at 30 uMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 169nMAssay Description:The opioid activity against the mu-receptor in the isolated guinea pig ileum(GPI)More data for this Ligand-Target Pair