BDBM50002009 5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-indole::CHEMBL273235

SMILES Fc1ccc(cc1)-n1cc(C2CCNCC2)c2cc(Cl)ccc12

InChI Key InChIKey=YCXCLZSLZGBCTA-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50002009   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tcg Lifesciences

Curated by ChEMBL
LigandPNGBDBM50002009(5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-i...)
Affinity DataIC50:  204nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002009(5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-i...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tcg Lifesciences

Curated by ChEMBL
LigandPNGBDBM50002009(5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-i...)
Affinity DataIC50:  204nMAssay Description:Inhibition of K+ channel activity in CHO cells expressing HERG Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002009(5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-i...)
Affinity DataIC50:  23nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed