BDBM50002310 3-[2-(Phenethyl-propyl-amino)-ethyl]-phenol; hydrobromide::CHEMBL1188090::CHEMBL545783
SMILES CCCN(CCc1ccccc1)CCc1cccc(O)c1
InChI Key InChIKey=QUZUPTMNMJTYGL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50002310
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]YM-09151-2 from human dopamine D3 receptor expressed in CHOp cellsMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Displacement of [3H]YM-09151-2 from human dopamine D2 receptor expressed in CHOp cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.71E+3nMAssay Description:Displacement of [3H]pCl-DPDPE from human delta opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH-23390 from human dopamine D1 receptor expressed in LHD1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cell membranes incubated for 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]ethylketocyclazocine from kappa opioid receptor in guinea pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at human dopamine D2 receptor expressed in CHOp cells assessed as stimulation of mitogenesis incubated for 24 hrs by [3H]thymidine i...More data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHOp cells assessed as stimulation of mitogenesis incubated for 24 hrs by [3H]thymidine i...More data for this Ligand-Target Pair
Affinity DataIC50: 9.28E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair