BDBM50010659 CHEMBL3264748
SMILES [H][C@]12O[C@]34CC[C@@]5(OCOc6c(O)ccc7C[C@@]3([H])N(CC3CC3)CC[C@]4(c67)[C@]15[H])N(CCc1ccccc1)C2=O
InChI Key InChIKey=ASWPFFLMSHOYIM-NLIGWKNISA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50010659
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
Affinity DataEC50: 0.620nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at human kappa opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 0.410nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair