BDBM50014091 CHEMBL3260847

SMILES CC(C)(C)NC(=O)C(N(Cc1ccccc1)C=O)c1c([nH]c2cc(Cl)ccc12)C(O)=O

InChI Key InChIKey=ZINAJZLZQYEGQO-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50014091   

TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50014091(CHEMBL3260847)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from human recombinant N-terminal domain of MDM2 (1 to 118 residues) expressed in Escherichia coli BL21 (DE3) cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50014091(CHEMBL3260847)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of fluorescent P4 peptide from MDM2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed