BDBM50019818 7-Chloro-3-naphthalen-2-ylmethyl-5-phenyl-1,3-dihydro-benzo[e][1,4]diazepin-2-one::CHEMBL20514

SMILES Clc1ccc2NC(=O)C(Cc3ccc4ccccc4c3)N=C(c3ccccc3)c2c1

InChI Key InChIKey=DJLHFAWVRFCKPO-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50019818   

TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50019818(7-Chloro-3-naphthalen-2-ylmethyl-5-phenyl-1,3-dihy...)
Affinity DataIC50:  6.10E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019818(7-Chloro-3-naphthalen-2-ylmethyl-5-phenyl-1,3-dihy...)
Affinity DataIC50:  4.90E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019818(7-Chloro-3-naphthalen-2-ylmethyl-5-phenyl-1,3-dihy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed