BDBM50026968 9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-benzo[d]pyrrolo[1,2-a]azepine::CHEMBL415761

SMILES [#6]-[#7]-1-[#6]-[#6]\[#6](-[#6]-[#6]-1)=[#6]-1/c2cccn2-[#6]=[#6]-c2ccc(Cl)cc-12

InChI Key InChIKey=VKQBOOLQCCBQAZ-UHFFFAOYSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50026968   

TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]- clonidine radioligand binding at the alpha-2 adrenergic receptor binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed