BDBM50042712 10-(2-Methyl-imidazol-1-ylmethyl)-5,6,9,10-tetrahydro-4H,8H-pyrido[3,2,1-jk]carbazol-11-one::CHEMBL332242

SMILES Cc1nccn1CC1CCc2c(C1=O)c1cccc3CCCn2c13

InChI Key InChIKey=NCNFDKWULDWJDS-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50042712   

Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Solvay Duphar

Curated by ChEMBL
LigandPNGBDBM50042712(10-(2-Methyl-imidazol-1-ylmethyl)-5,6,9,10-tetrahy...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Solvay Duphar

Curated by ChEMBL
LigandPNGBDBM50042712(10-(2-Methyl-imidazol-1-ylmethyl)-5,6,9,10-tetrahy...)
Affinity DataKi:  1.10nMAssay Description:The binding affinity of the compound was measured on mu-opiate receptor using [3H]- naloxone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Solvay Duphar

Curated by ChEMBL
LigandPNGBDBM50042712(10-(2-Methyl-imidazol-1-ylmethyl)-5,6,9,10-tetrahy...)
Affinity DataKi:  1.10nMAssay Description:The binding affinity of the compound was measured on kappa-opiate receptor using [3H]- EKC as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed