BDBM50060137 (1R,2S)-4-aminocyclopentane-1,2,4-tricarboxylic acid::(1R,2S,4s)-4-aminocyclopentane-1,2,4-tricarboxylic acid::(1S,2R,4S)-4-Amino-cyclopentane-1,2,4-tricarboxylic acid::(1S,2R,4s)-4-aminocyclopentane-1,2,4-tricarboxylic acid::4-Amino-cyclopentane-1,2,4-tricarboxylic acid::CHEMBL285043
SMILES N[C@]1(C[C@@H]([C@@H](C1)C(O)=O)C(O)=O)C(O)=O
InChI Key InChIKey=FERIKTBTNCSGJS-KIGHRTHISA-N
Data 16 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 16 hits for monomerid = 50060137
Affinity DataEC50: 7.20E+3nMAssay Description:Agonist activity against Metabotropic glutamate receptor 4 expressed in HEK 293 cells was evaluated by measuring total inositol phosphate accumulatio...More data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat mGluR2 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 7.20E+3nMAssay Description:Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.20E+6nMAssay Description:Activity at rat mGluR7 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat mGluR5 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.01E+4nMAssay Description:Activity at rat mGluR8 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.84E+4nMAssay Description:Activity at rat mGluR6 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 2.80E+5nMAssay Description:Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Faust Pharmaceuticals
Curated by ChEMBL
Faust Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 1.06E+4nMAssay Description:Agonist activity at rat mGlu6 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+5nMAssay Description:Agonist activity at mGlu7 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+3nMAssay Description:Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assayMore data for this Ligand-Target Pair