BDBM50062279 CHEMBL416789::Phosphoric acid mono-[5-(6-amino-purin-9-yl)-4-hydroxy-2-phosphonooxymethyl-tetrahydro-furan-3-yl] ester::US11185100, TABLE 7.1
SMILES Nc1ncnc2n(cnc12)C1OC(COP(O)(O)=O)C(OP(O)(O)=O)C1O
InChI Key InChIKey=WHTCPDAXWFLDIH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 50062279
Affinity DataIC50: 4.19E+3nMAssay Description:Antagonist activity at P2Y1 receptor measured as capacity to inhibit 50% of phospholipase C stimulation elicited by 10 nM 2-MeSATPMore data for this Ligand-Target Pair
Affinity DataEC50: 1.28E+3nMAssay Description:Agonist activity at P2Y1 receptor measured as capacity to stimulate 50% phospholipase C in turkey erythrocyte membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+4nMAssay Description:In vitro antagonist activity at P2Y1 receptor in turkey erythrocyte membranes.More data for this Ligand-Target Pair
Affinity DataEC50: 2.34E+3nMAssay Description:Concentration at which 50% of the maximal effect (stimulation of PLC at P2Y1 receptor in the turkey erythrocyte membranes) is reachedMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:The concentration of alanine is 20 mM.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:HEK293 cells that stably express T1R3 and inducibly express T1R1 were exposed to nucleotide derivatives alone to activate the umami receptor. Activat...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:The concentration of alanine is 20 mM.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The concentration of IMP is 0.2 mM.More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:HEK293 cells that stably express T1R3 and inducibly express T1R1 were exposed to nucleotide derivatives alone to activate the umami receptor. Activat...More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:The concentration of alanine is 20 mM.More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:HEK293 cells that stably express T1R3 and inducibly express T1R1 were exposed to nucleotide derivatives alone to activate the umami receptor. Activat...More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:The concentration of alanine is 20 mM.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The concentration of alanine is 20 mM.More data for this Ligand-Target Pair